Immunotherapy Drugs 🛡️

⚠️ Important Safety Notes

  • Immunotherapy can cause immune-related adverse events (irAEs) - monitor closely
  • Side effects can occur weeks to months after treatment - long-term monitoring required
  • Many side effects are reversible with early recognition and treatment
  • Always consult oncology team for any suspected immune-related toxicity
  • Steroids are often first-line treatment for moderate-severe irAEs

🔬 How Immunotherapy Works

  • Checkpoint inhibitors block proteins that prevent immune system from attacking cancer cells
  • PD-1/PD-L1 inhibitors: Block interaction between cancer cells and T-cells
  • CTLA-4 inhibitors: Enhance T-cell activation and proliferation
  • Monoclonal antibodies: Target specific proteins on cancer cells
  • CAR-T therapy: Genetically modified T-cells to recognize cancer antigens

Common Immune-Related Adverse Events (irAEs)

  • Skin: Rash, pruritus, vitiligo, Stevens-Johnson syndrome
  • GI: Diarrhea, colitis, hepatitis, pancreatitis
  • Endocrine: Thyroid dysfunction, diabetes, adrenal insufficiency
  • Pulmonary: Pneumonitis, interstitial lung disease
  • Neurological: Neuropathy, encephalitis, myasthenia gravis
  • Cardiac: Myocarditis, pericarditis, arrhythmias
  • Renal: Nephritis, acute kidney injury

Monitoring Requirements

  • Baseline: FBC, U&E, LFTs, TFTs, cortisol, glucose, CXR
  • During treatment: FBC, U&E, LFTs every 2-4 weeks
  • TFTs every 6-8 weeks (more frequent if symptoms)
  • Chest imaging if respiratory symptoms develop
  • Cardiac monitoring if cardiac symptoms
  • Skin examination at each visit

Emergency Management

  • Severe diarrhea (>6 stools/day): Stop immunotherapy, start high-dose steroids
  • Pneumonitis: Stop immunotherapy, high-dose steroids, consider antibiotics
  • Hepatitis (ALT >3x ULN): Stop immunotherapy, high-dose steroids
  • Myocarditis: Stop immunotherapy, cardiology review, high-dose steroids
  • Stevens-Johnson syndrome: Stop immunotherapy, dermatology review, high-dose steroids
  • Adrenal crisis: Hydrocortisone 100mg IV, endocrinology review

Pre-treatment Assessment

  • Full blood count, renal and liver function
  • Thyroid function tests and cortisol levels
  • Baseline chest X-ray or CT
  • ECG and echo if cardiac risk factors
  • Autoimmune disease history (relative contraindication)
  • Performance status assessment
  • Baseline skin examination

🔗 Related Topics

🛡️Immunotherapy Drugs Reference

Pembrolizumab
PD-1
Dose:200mg IV every 3 weeks
Indication:Melanoma, NSCLC, HNSCC, RCC, MSI-H cancers
Side Effects: Fatigue, rash, diarrhea, pneumonitis, thyroid dysfunction
Monitoring: FBC, U&E, LFTs, TFTs, CXR
Nivolumab
PD-1
Dose:240mg IV every 2 weeks
Indication:Melanoma, NSCLC, RCC, HNSCC, HCC
Side Effects: Fatigue, rash, diarrhea, pneumonitis, thyroid dysfunction
Monitoring: FBC, U&E, LFTs, TFTs, CXR
Atezolizumab
PD-L1
Dose:840mg IV every 2 weeks
Indication:NSCLC, SCLC, urothelial carcinoma, triple-negative breast cancer
Side Effects: Fatigue, rash, diarrhea, pneumonitis, thyroid dysfunction
Monitoring: FBC, U&E, LFTs, TFTs, CXR
Durvalumab
PD-L1
Dose:10mg/kg IV every 2 weeks
Indication:NSCLC, urothelial carcinoma
Side Effects: Fatigue, rash, diarrhea, pneumonitis, thyroid dysfunction
Monitoring: FBC, U&E, LFTs, TFTs, CXR
Ipilimumab
CTLA-4
Dose:3mg/kg IV every 3 weeks
Indication:Melanoma, RCC (in combination)
Side Effects: Diarrhea, colitis, hepatitis, rash, hypophysitis
Monitoring: FBC, U&E, LFTs, TFTs, cortisol
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Important Safety Notes

Immunotherapy can cause immune-related adverse events (irAEs) that may occur weeks to months after treatment. Early recognition and treatment are crucial. Always consult the oncology team for any suspected immune-related toxicity.